Publications (46) Publications in which a researcher has participated

filter_list Drug Discovery

2024

  1. 1,2,3-Triazole-totarol conjugates as potent PIP5K1α lipid kinase inhibitors

    Bioorganic and Medicinal Chemistry, Vol. 105

  2. A one-pot and eco-friendly synthesis of novel β-substituted-α-halomethyl acrylates and the bioactivity of these compounds in an in vitro model of mast cell degranulation induced by pro-inflammatory stimuli

    Biomedicine and Pharmacotherapy, Vol. 170

  3. Synthesis, Biological Activity, and Molecular-Docking Studies of New Brassinosteroid Analogs

    International Journal of Molecular Sciences, Vol. 25, Núm. 18

2023

  1. Labdane conjugates protect cardiomyocytes from doxorubicin-induced cardiotoxicity

    Drug Development Research, Vol. 84, Núm. 1, pp. 84-95

  2. Methyl esters of 23,24-Dinor-5α-cholan-22-oic acids as brassinosteroid Analogues. Synthesis, evaluation of plant growth promoting activity and Molecular docking

    Steroids, Vol. 196

  3. Phenolic and quinone methide nor-triterpenes as selective NLRP3 inflammasome inhibitors

    Bioorganic Chemistry, Vol. 132

  4. Synthesis and biological evaluation of anthracene-9,10 dione derivatives as CK2 inhibitors

    Results in Chemistry, Vol. 6

  5. Synthesis of Structurally Related Coumarin Derivatives as Antiproliferative Agents

    ACS Omega, Vol. 8, Núm. 29, pp. 26479-26496

2022

  1. Dehydroisohispanolone as a Promising NLRP3 Inhibitor Agent: Bioevaluation and Molecular Docking

    Pharmaceuticals, Vol. 15, Núm. 7

  2. Design, Semisynthesis, and Estrogenic Activity of Lignan Derivatives from Natural Dibenzylbutyrolactones

    Pharmaceuticals, Vol. 15, Núm. 5, pp. 585

  3. Guanidine Derivatives Containing the Chalcone Skeleton Are Potent Antiproliferative Compounds against Human Leukemia Cells

    International journal of molecular sciences, Vol. 23, Núm. 24

  4. Structure-activity relationships reveal a 2-furoyloxychalcone as a potent cytotoxic and apoptosis inducer for human U-937 and HL-60 leukaemia cells

    Bioorganic Chemistry, Vol. 127

2020

  1. Dehydrohispanolone Derivatives Attenuate the Inflammatory Response through the Modulation of Inflammasome Activation

    Journal of Natural Products, Vol. 83, Núm. 7, pp. 2155-2164

  2. Design, synthesis and biological evaluation of new embelin derivatives as CK2 inhibitors

    Bioorganic Chemistry, Vol. 95

  3. Development of an in vitro screening assay for PIP5K1α lipid kinase and identification of potent inhibitors

    FEBS Journal, Vol. 287, Núm. 14, pp. 3042-3064

  4. The synthetic flavanone 6-methoxy-2-(naphthalen-1-yl)chroman-4-one induces apoptosis and activation of the MAPK pathway in human U-937 leukaemia cells

    Bioorganic Chemistry, Vol. 94

2019

  1. Metal complexes of natural product like-compounds with antitumor activity

    Anti-Cancer Agents in Medicinal Chemistry, Vol. 19, Núm. 1, pp. 48-65

2018

  1. A new family of densely functionalized fused-benzoquinones as potent human protein kinase CK2 inhibitors

    European Journal of Medicinal Chemistry, Vol. 144, pp. 410-423

  2. Semisynthesis and inhibitory effects of solidagenone derivatives on TLR-mediated inflammatory responses

    Molecules, Vol. 23, Núm. 12

2017

  1. 5-Ethynylarylnaphthalimides as antitumor agents: Synthesis and biological evaluation

    Bioorganic and Medicinal Chemistry, Vol. 25, Núm. 6, pp. 1976-1983