Publications (38) Publications in which a researcher has participated

filter_list Pharmacology

2024

  1. 1,2,3-Triazole-totarol conjugates as potent PIP5K1α lipid kinase inhibitors

    Bioorganic and Medicinal Chemistry, Vol. 105

  2. A one-pot and eco-friendly synthesis of novel β-substituted-α-halomethyl acrylates and the bioactivity of these compounds in an in vitro model of mast cell degranulation induced by pro-inflammatory stimuli

    Biomedicine and Pharmacotherapy, Vol. 170

  3. Synthesis, Biological Activity, and Molecular-Docking Studies of New Brassinosteroid Analogs

    International Journal of Molecular Sciences, Vol. 25, Núm. 18

2023

  1. Labdane conjugates protect cardiomyocytes from doxorubicin-induced cardiotoxicity

    Drug Development Research, Vol. 84, Núm. 1, pp. 84-95

  2. Phenolic and quinone methide nor-triterpenes as selective NLRP3 inflammasome inhibitors

    Bioorganic Chemistry, Vol. 132

  3. Synthesis and biological evaluation of anthracene-9,10 dione derivatives as CK2 inhibitors

    Results in Chemistry, Vol. 6

  4. Synthesis of Structurally Related Coumarin Derivatives as Antiproliferative Agents

    ACS Omega, Vol. 8, Núm. 29, pp. 26479-26496

2022

  1. Dehydroisohispanolone as a Promising NLRP3 Inhibitor Agent: Bioevaluation and Molecular Docking

    Pharmaceuticals, Vol. 15, Núm. 7

  2. Design, Semisynthesis, and Estrogenic Activity of Lignan Derivatives from Natural Dibenzylbutyrolactones

    Pharmaceuticals, Vol. 15, Núm. 5, pp. 585

  3. Structure-activity relationships reveal a 2-furoyloxychalcone as a potent cytotoxic and apoptosis inducer for human U-937 and HL-60 leukaemia cells

    Bioorganic Chemistry, Vol. 127

2021

  1. Autodisplay of human PIP5K1α lipid kinase on Escherichia coli and inhibitor testing

    Enzyme and Microbial Technology, Vol. 143

2020

  1. Dehydrohispanolone Derivatives Attenuate the Inflammatory Response through the Modulation of Inflammasome Activation

    Journal of Natural Products, Vol. 83, Núm. 7, pp. 2155-2164

  2. Development of an in vitro screening assay for PIP5K1α lipid kinase and identification of potent inhibitors

    FEBS Journal, Vol. 287, Núm. 14, pp. 3042-3064

  3. The synthetic flavanone 6-methoxy-2-(naphthalen-1-yl)chroman-4-one induces apoptosis and activation of the MAPK pathway in human U-937 leukaemia cells

    Bioorganic Chemistry, Vol. 94

2018

  1. 3′-Hydroxy-3,4′-dimethoxyflavone-induced cell death in human leukaemia cells is dependent on caspases and reactive oxygen species and attenuated by the inhibition of JNK/SAPK

    Chemico-Biological Interactions, Vol. 288, pp. 1-11

  2. Semisynthesis and inhibitory effects of solidagenone derivatives on TLR-mediated inflammatory responses

    Molecules, Vol. 23, Núm. 12

2017

  1. 3′-Hydroxy-3,4′-dimethoxyflavone blocks tubulin polymerization and is a potent apoptotic inducer in human SK-MEL-1 melanoma cells

    Bioorganic and Medicinal Chemistry, Vol. 25, Núm. 21, pp. 6060-6070

  2. Synthesis and biological evaluation of naphthoquinone-coumarin conjugates as topoisomerase II inhibitors

    Bioorganic and Medicinal Chemistry Letters, Vol. 27, Núm. 3, pp. 484-489

2015

  1. A new iridoid, verbascoside and derivatives with inhibitory activity against Taq DNA polymerase

    Bioorganic and Medicinal Chemistry Letters, Vol. 25, Núm. 4, pp. 914-918

  2. Antiproliferative and structure activity relationships of amaryllidaceae alkaloids

    Molecules, Vol. 20, Núm. 8, pp. 13854-13863