![Foto de Ángel Ernesto](/img/nophoto.png)
Ángel Ernesto
Amesty Arrieta
Investigador en el període 2016-2023
Publicacions (35) Publicacions de Ángel Ernesto Amesty Arrieta
2024
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1,2,3-Triazole-totarol conjugates as potent PIP5K1α lipid kinase inhibitors
Bioorganic and Medicinal Chemistry, Vol. 105
2023
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Labdane conjugates protect cardiomyocytes from doxorubicin-induced cardiotoxicity
Drug Development Research, Vol. 84, Núm. 1, pp. 84-95
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Methyl esters of 23,24-Dinor-5α-cholan-22-oic acids as brassinosteroid Analogues. Synthesis, evaluation of plant growth promoting activity and Molecular docking
Steroids, Vol. 196
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Phenolic and quinone methide nor-triterpenes as selective NLRP3 inflammasome inhibitors
Bioorganic Chemistry, Vol. 132
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Synthesis and biological evaluation of anthracene-9,10 dione derivatives as CK2 inhibitors
Results in Chemistry, Vol. 6
2022
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Dehydroisohispanolone as a Promising NLRP3 Inhibitor Agent: Bioevaluation and Molecular Docking
Pharmaceuticals, Vol. 15, Núm. 7
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Design, Semisynthesis, and Estrogenic Activity of Lignan Derivatives from Natural Dibenzylbutyrolactones
Pharmaceuticals, Vol. 15, Núm. 5, pp. 585
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Discovery of Highly Functionalized 5-hydroxy-2H-pyrrol-2-ones That Exhibit Antiestrogenic Effects in Breast and Endometrial Cancer Cells and Potentiate the Antitumoral Effect of Tamoxifen
Cancers, Vol. 14, Núm. 21
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Flavonoids from Piper Species as Promising Antiprotozoal Agents against Giardia intestinalis: Structure-Activity Relationship and Drug-Likeness Studies
Pharmaceuticals, Vol. 15, Núm. 11
2021
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JKST6, a novel multikinase modulator of the BCR-ABL1/STAT5 signaling pathway that potentiates direct BCR-ABL1 inhibition and overcomes imatinib resistance in chronic myelogenous leukemia
Biomedicine and Pharmacotherapy, Vol. 144
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Modular synthesis and antiproliferative activity of new dihydro-1H-pyrazolo[1,3-b]pyridine embelin derivatives
Pharmaceuticals, Vol. 14, Núm. 10
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Synthesis and fungicidal activity of hydrated geranylated phenols against botrytis cinerea
Molecules, Vol. 26, Núm. 22
2020
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Dehydrohispanolone Derivatives Attenuate the Inflammatory Response through the Modulation of Inflammasome Activation
Journal of Natural Products, Vol. 83, Núm. 7, pp. 2155-2164
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Design, synthesis and biological evaluation of new embelin derivatives as CK2 inhibitors
Bioorganic Chemistry, Vol. 95
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Development of an in vitro screening assay for PIP5K1α lipid kinase and identification of potent inhibitors
FEBS Journal, Vol. 287, Núm. 14, pp. 3042-3064
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Efficient Multicomponent Synthesis of Diverse Antibacterial Embelin-Privileged Structure Conjugates
Molecules (Basel, Switzerland), Vol. 25, Núm. 14
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Withanolide-Type Steroids from Withania aristata as Potential Anti-Leukemic Agents
Molecules (Basel, Switzerland), Vol. 25, Núm. 23
2019
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A novel naphthoquinone-coumarin hybrid that inhibits BCR-ABL1-STAT5 oncogenic pathway and reduces survival in imatinib-resistant chronic myelogenous leukemia cells
Frontiers in Pharmacology, Vol. 9, Núm. JAN
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Expanding the Chemical Space of Withaferin A by Incorporating Silicon to Improve Its Clinical Potential on Human Ovarian Carcinoma Cells
Journal of Medicinal Chemistry, Vol. 62, Núm. 9, pp. 4571-4585
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Metal complexes of natural product like-compounds with antitumor activity
Anti-Cancer Agents in Medicinal Chemistry, Vol. 19, Núm. 1, pp. 48-65