Publicaciones (44) Publicaciones de Adrián Puerta Arocha

2024

  1. Coumarins-lipophilic cations conjugates: Efficient mitocans targeting carbonic anhydrases

    Bioorganic Chemistry, Vol. 145

  2. Early pharmacological profiling of isatin derivatives as potent and selective cytotoxic agents

    Biochemical Pharmacology, Vol. 222

  3. Microwave-induced one-pot synthesis of 3-imidazolyl indole clubbed 1,2,3-triazole hybrids as antiproliferative agents and density functional theory study

    Archiv der Pharmazie, Vol. 357, Núm. 3

2023

  1. Antiproliferative effect of natural and semisynthetic polyethers from Laurencia viridis

    Natural Product Research

  2. Biotinylated selenocyanates: Potent and selective cytostatic agents

    Bioorganic Chemistry, Vol. 133

  3. Conformationally Restricted Glycoconjugates Derived from Arylsulfonamides and Coumarins: New Families of Tumour-Associated Carbonic Anhydrase Inhibitors

    International Journal of Molecular Sciences, Vol. 24, Núm. 11

  4. Fluoro-labelled sp2-iminoglycolipids with immunomodulatory properties

    European Journal of Medicinal Chemistry, Vol. 255

  5. Insights into microwave assisted synthesis of spiro-chromeno[2,3-d]pyrimidines using PEG-OSO3H catalyst: DFT study and their antiproliferative activity

    Journal of Molecular Structure, Vol. 1292

  6. Investigation of the enantioselectivity of acetylcholinesterase and butyrylcholinesterase upon inhibition by tacrine-iminosugar heterodimers

    Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 38, Núm. 1, pp. 349-360

  7. N-Substituted 3-Aminooxindoles and N-Propargyl Derivatives: Potential Biological Activities against Alzheimer's Disease

    Results in Chemistry, Vol. 6

  8. Structural, physicochemical and anticancer study of Zn complexes with pyridyl-based thiazolyl-hydrazones

    Journal of Molecular Structure, Vol. 1281

  9. Synthesis, antiproliferative evaluation and in silico studies of a novel steroidal spiro morpholinone

    Steroids, Vol. 192

  10. Tetranuclear Ru2Cu2 and Ru2Ni2 complexes with nanomolar anticancer activity

    Dalton Transactions, Vol. 52, Núm. 28, pp. 9541-9545

2022

  1. 2-Aminobenzoxazole-appended coumarins as potent and selective inhibitors of tumour-associated carbonic anhydrases

    Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 37, Núm. 1, pp. 168-177

  2. A Comprehensive Evaluation of Sdox, a Promising H2S-Releasing Doxorubicin for the Treatment of Chemoresistant Tumors

    Frontiers in Pharmacology, Vol. 13

  3. A hybrid of 1-deoxynojirimycin and benzotriazole induces preferential inhibition of butyrylcholinesterase (BuChE) over acetylcholinesterase (AChE)

    Journal of enzyme inhibition and medicinal chemistry, Vol. 37, Núm. 1, pp. 2395-2402

  4. A new oxadiazole-based topsentin derivative modulates cyclin-dependent kinase 1 expression and exerts cytotoxic effects on pancreatic cancer cells

    Molecules, Vol. 27, Núm. 1

  5. Alkaloid Profiling, Anti-Enzymatic and Antiproliferative Activity of the Endemic Chilean Amaryllidaceae Phycella cyrtanthoides

    Metabolites, Vol. 12, Núm. 2

  6. Bioactive Potential: A Pharmacognostic Definition through the Screening of Four Hypericum Species from the Canary Islands

    Molecules, Vol. 27, Núm. 18

  7. Carbohydrate-derived bicyclic selenazolines as new dual inhibitors (cholinesterases/OGA) against Alzheimer's disease

    Bioorganic Chemistry, Vol. 127