Instituto Universitario de Tecnologías Biomédicas
Institut de recherche
Instituto Canario de Investigación del Cáncer
Santa Cruz de Tenerife, EspañaPublications en collaboration avec des chercheurs de Instituto Canario de Investigación del Cáncer (33)
2014
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Yeast cytotoxic sensitivity to the antitumour agent β-lapachone depends mainly on oxidative stress and is largely independent of microtubule- or topoisomerase-mediated DNA damage
Biochemical Pharmacology, Vol. 92, Núm. 2, pp. 206-219
2013
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Achyrofuran is an antibacterial agent capable of killing methicillin-resistant vancomycin-intermediate Staphylococcus aureus in the nanomolar range
Phytomedicine, Vol. 20, Núm. 2, pp. 133-138
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Multicomponent synthesis of antibacterial dihydropyridin and dihydropyran embelin derivatives
Journal of Organic Chemistry, Vol. 78, Núm. 16, pp. 7977-7985
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Synthesis and study of antiproliferative, antitopoisomerase II, DNA-intercalating and DNA-damaging activities of arylnaphthalimides
Bioorganic and Medicinal Chemistry, Vol. 21, Núm. 21, pp. 6484-6495
2012
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Antiproliferative activity of withanolide derivatives from Jaborosa cabrerae and Jaborosa reflexa. Chemotaxonomic considerations
Phytochemistry, Vol. 76, pp. 150-157
2011
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Comparative analysis of the ERα/ERβ ratio and neurotensin and its high-affinity receptor in myometrium, uterine leiomyoma, atypical leiomyoma, and leiomyosarcoma
International Journal of Gynecological Pathology, Vol. 30, Núm. 4, pp. 354-363
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Neurotensina y otros Péptidos reguladores en el desarrollo hipofisario humano y en adenomas hipofisarios
BioCancer Research Journal, Vol. 5, pp. 161-170
2010
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Antiproliferative activity of novel benzo[b][1,6]naphthyridines in human solid tumor cell lines
Bioorganic and Medicinal Chemistry Letters, Vol. 20, Núm. 5, pp. 1504-1506
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Antiproliferative activity of synthetic naphthoquinones related to lapachol. First synthesis of 5-hydroxylapachol
Bioorganic and Medicinal Chemistry, Vol. 18, Núm. 7, pp. 2621-2630
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Enhancement of antiproliferative activity by molecular simplification of catalpol
Bioorganic and Medicinal Chemistry, Vol. 18, Núm. 7, pp. 2515-2523
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Mitotic arrest induced by a novel family of DNA topoisomerase II inhibitors
Journal of Medicinal Chemistry, Vol. 53, Núm. 9, pp. 3835-3839
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Neurotensin and neurotensin receptor 1 expression in human myometrium and uterine leiomyomas
Biology of Reproduction, Vol. 83, Núm. 4, pp. 641-647
2009
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Synthesis and antiproliferative activity of 2,4-disubstituted 6-aryl-7H-pyrrolo[3,2-d]pyrimidin-7-one 5-oxides
Bioorganic and Medicinal Chemistry, Vol. 17, Núm. 14, pp. 4955-4960
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Tessaric acid derivatives induce G2/M cell cycle arrest in human solid tumor cell lines
Bioorganic and Medicinal Chemistry, Vol. 17, Núm. 17, pp. 6251-6256
2008
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Design and synthesis of a novel series of pyranonaphthoquinones as topoisomerase II catalytic inhibitors
Journal of Medicinal Chemistry, Vol. 51, Núm. 21, pp. 6761-6772
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Expression of neurotensin and its receptors in pituitary adenomas
Journal of Neuroendocrinology, Vol. 20, Núm. 9, pp. 1052-1057
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β′-Hydroxy-α,β-unsaturated ketones: A new pharmacophore for the design of anticancer drugs. Part 2
ChemMedChem, Vol. 3, Núm. 11, pp. 1740-1747
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γ-Lactones α,β- and β,γ-fused to carbocycles as novel antiproliferative drugs
Bioorganic and Medicinal Chemistry Letters, Vol. 18, Núm. 19, pp. 5171-5173
2007
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Antiproliferative activity of 2-alkyl-4-halopiperidines and 2-alkyl-4-halo-1,2,5,6-tetrahydropyridines in solid tumor cell lines
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 10, pp. 2681-2684
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Antiproliferative activity of 4-chloro-5,6-dihydro-2H-pyrans. Part 2: Enhancement of drug cytotoxicity
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 11, pp. 3087-3090