José Manuel
Padrón Carrillo
Catedrático de Universidad
Instituto Canario de Investigación del Cáncer
Santa Cruz de Tenerife, EspañaPublicacions en col·laboració amb investigadors/es de Instituto Canario de Investigación del Cáncer (21)
2012
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Antiproliferative activity of withanolide derivatives from Jaborosa cabrerae and Jaborosa reflexa. Chemotaxonomic considerations
Phytochemistry, Vol. 76, pp. 150-157
2010
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Antiproliferative activity of novel benzo[b][1,6]naphthyridines in human solid tumor cell lines
Bioorganic and Medicinal Chemistry Letters, Vol. 20, Núm. 5, pp. 1504-1506
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Antiproliferative activity of synthetic naphthoquinones related to lapachol. First synthesis of 5-hydroxylapachol
Bioorganic and Medicinal Chemistry, Vol. 18, Núm. 7, pp. 2621-2630
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Enhancement of antiproliferative activity by molecular simplification of catalpol
Bioorganic and Medicinal Chemistry, Vol. 18, Núm. 7, pp. 2515-2523
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Mitotic arrest induced by a novel family of DNA topoisomerase II inhibitors
Journal of Medicinal Chemistry, Vol. 53, Núm. 9, pp. 3835-3839
2009
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Synthesis and antiproliferative activity of 2,4-disubstituted 6-aryl-7H-pyrrolo[3,2-d]pyrimidin-7-one 5-oxides
Bioorganic and Medicinal Chemistry, Vol. 17, Núm. 14, pp. 4955-4960
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Tessaric acid derivatives induce G2/M cell cycle arrest in human solid tumor cell lines
Bioorganic and Medicinal Chemistry, Vol. 17, Núm. 17, pp. 6251-6256
2008
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β′-Hydroxy-α,β-unsaturated ketones: A new pharmacophore for the design of anticancer drugs. Part 2
ChemMedChem, Vol. 3, Núm. 11, pp. 1740-1747
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γ-Lactones α,β- and β,γ-fused to carbocycles as novel antiproliferative drugs
Bioorganic and Medicinal Chemistry Letters, Vol. 18, Núm. 19, pp. 5171-5173
2007
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Antiproliferative activity of 2-alkyl-4-halopiperidines and 2-alkyl-4-halo-1,2,5,6-tetrahydropyridines in solid tumor cell lines
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 10, pp. 2681-2684
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Antiproliferative activity of 4-chloro-5,6-dihydro-2H-pyrans. Part 2: Enhancement of drug cytotoxicity
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 11, pp. 3087-3090
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Cytotoxic effects of C-glycosides in HOS and HeLa cell lines
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 13, pp. 3676-3681
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Inhibition of DNA topoisomerase I and growth inhibition of human cancer cell lines by an oleanane from Junellia aspera (Verbenaceae)
Cellular and Molecular Biology, Vol. 53, Núm. 3, pp. 13-17
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Novel antiproliferative analogs of the Taq DNA polymerase inhibitor catalpol
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 5, pp. 1332-1335
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Samarium(II) promoted stereoselective synthesis of antiproliferative cis-β-alkoxy-γ-alkyl-γ-lactones
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 1, pp. 18-21
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Synthesis and antiproliferative activity of (2R,3R)-disubstituted tetrahydropyrans. Part 2: Effect of side chain homologation
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 3, pp. 780-783
2006
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Abietane diterpenoids from Salvia pachyphylla and S. clevelandii with cytotoxic activity against human cancer cell lines
Journal of Natural Products, Vol. 69, Núm. 12, pp. 1803-1805
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Synthesis and antiproliferative activity of (2R,3R)-disubstituted tetrahydropyrans
Bioorganic and Medicinal Chemistry Letters, Vol. 16, Núm. 23, pp. 6135-6138
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Synthesis and antiproliferative activity of novel sugiol β-amino alcohol analogs
European Journal of Medicinal Chemistry, Vol. 41, Núm. 11, pp. 1327-1332
2005
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Antiproliferative activity in HL60 cells by tetrasubstituted pyrroles: A structure-activity relationship study
Bioorganic and Medicinal Chemistry Letters, Vol. 15, Núm. 10, pp. 2487-2490