José Manuel
Padrón Carrillo
Professeur Titulaire
Instituto Canario de Investigación del Cáncer
Santa Cruz de Tenerife, EspañaPublications en collaboration avec des chercheurs de Instituto Canario de Investigación del Cáncer (21)
2012
-
Antiproliferative activity of withanolide derivatives from Jaborosa cabrerae and Jaborosa reflexa. Chemotaxonomic considerations
Phytochemistry, Vol. 76, pp. 150-157
2010
-
Antiproliferative activity of novel benzo[b][1,6]naphthyridines in human solid tumor cell lines
Bioorganic and Medicinal Chemistry Letters, Vol. 20, Núm. 5, pp. 1504-1506
-
Antiproliferative activity of synthetic naphthoquinones related to lapachol. First synthesis of 5-hydroxylapachol
Bioorganic and Medicinal Chemistry, Vol. 18, Núm. 7, pp. 2621-2630
-
Enhancement of antiproliferative activity by molecular simplification of catalpol
Bioorganic and Medicinal Chemistry, Vol. 18, Núm. 7, pp. 2515-2523
-
Mitotic arrest induced by a novel family of DNA topoisomerase II inhibitors
Journal of Medicinal Chemistry, Vol. 53, Núm. 9, pp. 3835-3839
2009
-
Synthesis and antiproliferative activity of 2,4-disubstituted 6-aryl-7H-pyrrolo[3,2-d]pyrimidin-7-one 5-oxides
Bioorganic and Medicinal Chemistry, Vol. 17, Núm. 14, pp. 4955-4960
-
Tessaric acid derivatives induce G2/M cell cycle arrest in human solid tumor cell lines
Bioorganic and Medicinal Chemistry, Vol. 17, Núm. 17, pp. 6251-6256
2008
-
β′-Hydroxy-α,β-unsaturated ketones: A new pharmacophore for the design of anticancer drugs. Part 2
ChemMedChem, Vol. 3, Núm. 11, pp. 1740-1747
-
γ-Lactones α,β- and β,γ-fused to carbocycles as novel antiproliferative drugs
Bioorganic and Medicinal Chemistry Letters, Vol. 18, Núm. 19, pp. 5171-5173
2007
-
Antiproliferative activity of 2-alkyl-4-halopiperidines and 2-alkyl-4-halo-1,2,5,6-tetrahydropyridines in solid tumor cell lines
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 10, pp. 2681-2684
-
Antiproliferative activity of 4-chloro-5,6-dihydro-2H-pyrans. Part 2: Enhancement of drug cytotoxicity
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 11, pp. 3087-3090
-
Cytotoxic effects of C-glycosides in HOS and HeLa cell lines
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 13, pp. 3676-3681
-
Inhibition of DNA topoisomerase I and growth inhibition of human cancer cell lines by an oleanane from Junellia aspera (Verbenaceae)
Cellular and Molecular Biology, Vol. 53, Núm. 3, pp. 13-17
-
Novel antiproliferative analogs of the Taq DNA polymerase inhibitor catalpol
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 5, pp. 1332-1335
-
Samarium(II) promoted stereoselective synthesis of antiproliferative cis-β-alkoxy-γ-alkyl-γ-lactones
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 1, pp. 18-21
-
Synthesis and antiproliferative activity of (2R,3R)-disubstituted tetrahydropyrans. Part 2: Effect of side chain homologation
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 3, pp. 780-783
2006
-
Abietane diterpenoids from Salvia pachyphylla and S. clevelandii with cytotoxic activity against human cancer cell lines
Journal of Natural Products, Vol. 69, Núm. 12, pp. 1803-1805
-
Synthesis and antiproliferative activity of (2R,3R)-disubstituted tetrahydropyrans
Bioorganic and Medicinal Chemistry Letters, Vol. 16, Núm. 23, pp. 6135-6138
-
Synthesis and antiproliferative activity of novel sugiol β-amino alcohol analogs
European Journal of Medicinal Chemistry, Vol. 41, Núm. 11, pp. 1327-1332
2005
-
Antiproliferative activity in HL60 cells by tetrasubstituted pyrroles: A structure-activity relationship study
Bioorganic and Medicinal Chemistry Letters, Vol. 15, Núm. 10, pp. 2487-2490